Synlett

Synthesis of novel indole derivatives: variations in the Bartoli reaction

AP Dobbs, M Voyle, N Whittall

Index: Dobbs, Adrian P.; Voyle, Martyn; Whittall, Neil Synlett, 1999 , # 10 p. 1594 - 1596

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Citation Number: 18

Abstract

Adrian P. Dobbs,1* Martyn Voyle, Neil Whittall SmithKline Beecham Pharmaceuticals, Old Powder Mills, Leigh, Tonbridge, Kent TN11 9AN, UK E-mail: adrian@apdobbs.demon.co.uk; Neil_Whittall-1@sbphrd.com Received 29 June 1999 ... Abstract: The synthesis of a range of novel substituted indoles and tricyclic indole derivatives is described using an extension of the Bartoli methodology. Key words: Grignard reactions, indoles, Bartoli reaction, regiose- ...

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