117332-69-1

117332-69-1 structure

Name: Clocinnamox mesylate
Chemical Name: 14b-(p-chlorocinnamoylamino)-7,8-dihydro-n-cyclopropylmethylmorphinone mesylate
CAS Number: 117332-69-1
Molecular Formula: C₃₀H₃₃ClN₂O₇S
Molecular Weight: 601.11
Catalog: Organic raw materials Amino compound Sulfonic acid amino compound
Create Date: 2018-12-08 21:06:31
Modify Date: 2024-01-11 17:21:14
Clocinnamox (mesylate) is a potent opioid antagonist acting at mu, kappa and delta-receptors. Clocinnamox is a selective mu-receptor antagonist than kappa and delta-receptors[1].

Name	14b-(p-chlorocinnamoylamino)-7,8-dihydro-n-cyclopropylmethylmorphinone mesylate
Synonyms	clocinnamox threo Ifenprodil hemitartrate CLOCINNAMOX MESYLATE

Description	Clocinnamox (mesylate) is a potent opioid antagonist acting at mu, kappa and delta-receptors. Clocinnamox is a selective mu-receptor antagonist than kappa and delta-receptors[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Opioid Receptor Signaling Pathways >> Neuronal Signaling >> Opioid Receptor Research Areas >> Neurological Disease
References	[1]. S D Comer, et, al. Clocinnamox: a novel, systemically-active, irreversible opioid antagonist. J Pharmacol Exp Ther. 1992, 262, 3. [2]. E R Butelman, et, al. Clocinnamox antagonism of opioid suppression of schedule-controlled responding in rhesus monkeys. Psychopharmacology (Berl). 1996, 123, 4.