2219321-25-0

2219321-25-0 structure
2219321-25-0 structure
  • Name: GSK2973980A
  • Chemical Name: GSK2973980A
  • CAS Number: 2219321-25-0
  • Molecular Formula: C25H19F5N4O4
  • Molecular Weight: 534.43
  • Catalog: Signaling Pathways Metabolic Enzyme/Protease Acyltransferase
  • Create Date: 2019-03-30 20:49:34
  • Modify Date: 2024-01-05 16:58:37
  • GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.

Name GSK2973980A
Description GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.
Related Catalog
Target

IC50: 3 nM (DGAT1)[1]

References

[1]. Cheung M, et al. Discovery of Tetralones as Potent and Selective Inhibitors of Acyl-CoA:Diacylglycerol Acyltransferase 1. ACS Med Chem Lett. 2018 Jan 16;9(2):103-108.

Molecular Formula C25H19F5N4O4
Molecular Weight 534.43