Shanghai Nianxing Industrial Co., Ltd
China
Product Name: ZEN-3219
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1952264-34-4

1952264-34-4 structure

1952264-34-4 structure

Name: ZEN-3219
Chemical Name: ZEN-3219
CAS Number: 1952264-34-4
Molecular Formula: C₁₉H₁₈N₂O₃
Molecular Weight: 322.36
Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
Create Date: 2019-06-01 10:28:29
Modify Date: 2024-01-03 16:33:24
ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4[1].

Name	ZEN-3219

Description	ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
Target	BRD4 (BD1):0.48 μM (IC50) BRD4 (BD2):0.16 μM (IC50) BRD4(BD1BD2):0.47 μM (IC50)
References	[1]. Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211.

Molecular Formula	C₁₉H₁₈N₂O₃
Molecular Weight	322.36

Hazard Codes	Xi

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