2035912-55-9

2035912-55-9 structure

Name: LSD1-IN-5
Chemical Name: LSD1-IN-5
CAS Number: 2035912-55-9
Molecular Formula: C₁₅H₁₃BrN₂O₃
Molecular Weight: 349.18
Catalog: Signaling Pathways Epigenetics Histone Demethylase
Create Date: 2019-08-03 18:39:58
Modify Date: 2024-01-10 12:12:47
LSD1-IN-5 (Compound 4e) is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 121 nM. LSD1-IN-5 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1[1].

Name	LSD1-IN-5

Description	LSD1-IN-5 (Compound 4e) is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 121 nM. LSD1-IN-5 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Histone Demethylase
Target	IC50: 121 nM (LSD1)[1]
References	[1]. Duan YC, et al. Discovery of resveratrol derivatives as novel LSD1 inhibitors: Design, synthesis and their biological evaluation. Eur J Med Chem. 2017 Jan 27;126:246-258.

Molecular Formula	C₁₅H₁₃BrN₂O₃
Molecular Weight	349.18