Name | WRG-28 |
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Description | WRG-28 is a selective, extracellularly acting DDR2 allosteric inhibitor with an IC50 of 230 nM. WRG-28 uniquely inhibits receptor-ligand interactions via allosteric modulation of the receptor. WRG-28 inhibits tumor invasion and migration, as well as tumor-supporting roles of the stroma, and inhibits metastatic breast tumor cell colonization in the lungs by targeting DDR2[1]. |
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Related Catalog | |
Target |
DDR2:230 nM (IC50) |
References |
Molecular Formula | C21H18N2O5S |
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Molecular Weight | 410.44 |
Hazard Codes | Xi |
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