1217628-73-3
1217628-73-3 structure
- Name: SB 205607 dihydrobromide
- Chemical Name: 3-[(4aS,12aR)-2-Methyl-1,3,4,5,12,12a-hexahydropyrido[3,4-b]acridin-4a(2H)-yl]phenol dihydrobromide
- CAS Number: 1217628-73-3
- Molecular Formula: C23H24N2O.2HBr
- Molecular Weight: 506.273
- Catalog: Signaling Pathways GPCR/G Protein Opioid Receptor
- Create Date: 2020-01-11 14:33:41
- Modify Date: 2024-01-06 18:31:41
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A potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM; dispalys >1,000-fold selectivity over μOR and κOR; Pain Discontinued
| Name | 3-[(4aS,12aR)-2-Methyl-1,3,4,5,12,12a-hexahydropyrido[3,4-b]acridin-4a(2H)-yl]phenol dihydrobromide |
|---|---|
| Synonyms |
Phenol, 3-[(4aS,12aR)-1,3,4,5,12,12a-hexahydro-2-methylpyrido[3,4-b]acridin-4a(2H)-yl]-, hydrobromide (1:2)
3-[(4aS,12aR)-2-Methyl-1,3,4,5,12,12a-hexahydropyrido[3,4-b]acridin-4a(2H)-yl]phenol dihydrobromide |
| Description | A potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM; dispalys >1,000-fold selectivity over μOR and κOR; Pain Discontinued |
|---|---|
| References | References 1. Knapp RJ, et al. Eur J Pharmacol. 1995 Oct 15;291(2):129-34. 2. Tseng LF, et al. J Pharmacol Exp Ther. 1997 Feb;280(2):600-5. 3. Fusa K, et al. Neuroscience. 2005;130(3):745-55. View Related Products by Target Opioid Receptor Pain |
| Molecular Formula | C23H24N2O.2HBr |
|---|---|
| Molecular Weight | 506.273 |
| Exact Mass | 504.041168 |