SB 205607 dihydrobromide

Modify Date: 2024-01-06 18:31:41

SB 205607 dihydrobromide Structure
SB 205607 dihydrobromide structure
Common Name SB 205607 dihydrobromide
CAS Number 1217628-73-3 Molecular Weight 506.273
Density N/A Boiling Point N/A
Molecular Formula C23H24N2O.2HBr Melting Point N/A
MSDS N/A Flash Point N/A

 Use of SB 205607 dihydrobromide


A potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM; dispalys >1,000-fold selectivity over μOR and κOR; Pain Discontinued

 Names

Name 3-[(4aS,12aR)-2-Methyl-1,3,4,5,12,12a-hexahydropyrido[3,4-b]acridin-4a(2H)-yl]phenol dihydrobromide
Synonym More Synonyms

 SB 205607 dihydrobromide Biological Activity

Description A potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM; dispalys >1,000-fold selectivity over μOR and κOR; Pain Discontinued
References References 1. Knapp RJ, et al. Eur J Pharmacol. 1995 Oct 15;291(2):129-34. 2. Tseng LF, et al. J Pharmacol Exp Ther. 1997 Feb;280(2):600-5. 3. Fusa K, et al. Neuroscience. 2005;130(3):745-55. View Related Products by Target Opioid Receptor Pain

 Chemical & Physical Properties

Molecular Formula C23H24N2O.2HBr
Molecular Weight 506.273
Exact Mass 504.041168

 Synonyms

Phenol, 3-[(4aS,12aR)-1,3,4,5,12,12a-hexahydro-2-methylpyrido[3,4-b]acridin-4a(2H)-yl]-, hydrobromide (1:2)
3-[(4aS,12aR)-2-Methyl-1,3,4,5,12,12a-hexahydropyrido[3,4-b]acridin-4a(2H)-yl]phenol dihydrobromide