1802226-87-4
1802226-87-4 structure
- Name: PSB-12431
- Chemical Name: PSB-12431
- CAS Number: 1802226-87-4
- Molecular Formula: C18H22N4O10P2
- Molecular Weight: 516.34
- Create Date: 2020-01-19 23:15:57
- Modify Date: 2024-08-09 12:42:53
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PSB-12431 is an α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 9.2 nM for rat recombinant eN; displays high selectivity versus other ecto-nucleotidases and ADP-activated P2Y receptors, has high metabolic stability.
| Name | PSB-12431 |
|---|
| Description | PSB-12431 is an α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 9.2 nM for rat recombinant eN; displays high selectivity versus other ecto-nucleotidases and ADP-activated P2Y receptors, has high metabolic stability. |
|---|---|
| References | References 1. Bhattarai S, et al. J Med Chem. 2015 Aug 13;58(15):6248-63. View Related Products by Target Other Targets |
| Molecular Formula | C18H22N4O10P2 |
|---|---|
| Molecular Weight | 516.34 |