Name | BRD-IN-26 |
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Description | BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively; displays excellent selectivity over other bromodomains. |
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References | References 1. Sutherell CL, et al. J Med Chem. 2016 May 26;59(10):5095-101. View Related Products by Target Bromodomain |
Molecular Formula | C17H19ClN4O |
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Molecular Weight | 330.816 |