Name | TAK1-IN-1 |
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Description | TAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM, a thienopyrimidine scaffold that serves as a good starting point for medicinal chemistry. |
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References | References 1. Miura T, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):1031-1036. View Related Products by Target TAK1 |
Molecular Formula | C17H12N4O2S |
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Molecular Weight | 336.369 |