639863-77-7
639863-77-7 structure
- Name: N-Desmethyl Pimavanserin
- Chemical Name: N-Desmethyl Pimavanserin
- CAS Number: 639863-77-7
- Molecular Formula: C24H32FN3O2
- Molecular Weight: 413.53
- Create Date: 2020-01-23 13:15:51
- Modify Date: 2024-01-09 20:29:55
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N-Desmethyl Pimavanserin is the active metabolite of Pimavanserin. Pimavanserin is a selective inverse agonist of the 5-HT2A receptor with pIC50 and pKd of 8.73 and 9.3, respectively.
| Name | N-Desmethyl Pimavanserin |
|---|
| Description | N-Desmethyl Pimavanserin is the active metabolite of Pimavanserin. Pimavanserin is a selective inverse agonist of the 5-HT2A receptor with pIC50 and pKd of 8.73 and 9.3, respectively. |
|---|---|
| In Vitro | The mean plasma half-lives for Pimavanserin and its metabolite N-Desmethyl Pimavanserin (AC-279) are 57 hours and 200 hours, respectively. |
| References |
| Molecular Formula | C24H32FN3O2 |
|---|---|
| Molecular Weight | 413.53 |