N-Desmethyl Pimavanserin structure
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Common Name | N-Desmethyl Pimavanserin | ||
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CAS Number | 639863-77-7 | Molecular Weight | 413.53 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C24H32FN3O2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of N-Desmethyl PimavanserinN-Desmethyl Pimavanserin is the active metabolite of Pimavanserin. Pimavanserin is a selective inverse agonist of the 5-HT2A receptor with pIC50 and pKd of 8.73 and 9.3, respectively. |
Name | N-Desmethyl Pimavanserin |
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Description | N-Desmethyl Pimavanserin is the active metabolite of Pimavanserin. Pimavanserin is a selective inverse agonist of the 5-HT2A receptor with pIC50 and pKd of 8.73 and 9.3, respectively. |
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In Vitro | The mean plasma half-lives for Pimavanserin and its metabolite N-Desmethyl Pimavanserin (AC-279) are 57 hours and 200 hours, respectively. |
References |
Molecular Formula | C24H32FN3O2 |
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Molecular Weight | 413.53 |