Shanghai Nianxing Industrial Co., Ltd
China
Product Name: MCHR1 antagonist 3
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1069622-60-1

1069622-60-1 structure

1069622-60-1 structure

Name: MCHR1 antagonist 3
Chemical Name: MCHR1 antagonist 3
CAS Number: 1069622-60-1
Molecular Formula: C₂₉H₃₆N₄O₂
Molecular Weight: 472.62
Catalog: Signaling Pathways GPCR/G Protein MCHR1 (GPR24)
Create Date: 2020-06-01 09:34:55
Modify Date: 2025-08-20 09:27:58
MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism[1].

Name	MCHR1 antagonist 3

Description	MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism[1].
Related Catalog	Research Areas >> Endocrinology Signaling Pathways >> GPCR/G Protein >> MCHR1 (GPR24) Research Areas >> Metabolic Disease
In Vitro	Compound 1, derived from a spirohydantoin scaffold, exhibits a Ki of 50 nM at MCH-R1. Compound 1 is a potent inhibitor of CYP3A4 (IC50=35 nM). MCHR1 antagonist 3 is an analog of compound 1[1].
References	[1]. Rowbottom MW, et al. Synthesis and structure-activity relationships of spirohydantoin-derived small-moleculeantagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Bioorg Med Chem Lett. 2007 Apr 15;17(8):2171-8.

Molecular Formula	C₂₉H₃₆N₄O₂
Molecular Weight	472.62

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