MCHR1 antagonist 3

Modify Date: 2025-08-20 09:27:58

MCHR1 antagonist 3 Structure
MCHR1 antagonist 3 structure
Common Name MCHR1 antagonist 3
CAS Number 1069622-60-1 Molecular Weight 472.62
Density N/A Boiling Point N/A
Molecular Formula C29H36N4O2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of MCHR1 antagonist 3


MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism[1].

 Names

Name MCHR1 antagonist 3

 MCHR1 antagonist 3 Biological Activity

Description MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism[1].
Related Catalog
In Vitro Compound 1, derived from a spirohydantoin scaffold, exhibits a Ki of 50 nM at MCH-R1. Compound 1 is a potent inhibitor of CYP3A4 (IC50=35 nM). MCHR1 antagonist 3 is an analog of compound 1[1].
References

[1]. Rowbottom MW, et al. Synthesis and structure-activity relationships of spirohydantoin-derived small-moleculeantagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Bioorg Med Chem Lett. 2007 Apr 15;17(8):2171-8.

 Chemical & Physical Properties

Molecular Formula C29H36N4O2
Molecular Weight 472.62
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.