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299898-52-5

299898-52-5 structure
299898-52-5 structure
  • Name: (Pro3)-Gastric Inhibitory Polypeptide (human) trifluoroacetate salt
  • Chemical Name: (Pro3)-Gastric Inhibitory Polypeptide (human) trifluoroacetate salt
  • CAS Number: 299898-52-5
  • Molecular Formula: C226H338N60O64S
  • Molecular Weight:
  • Catalog: Signaling Pathways Protein Tyrosine Kinase/RTK Insulin Receptor
  • Create Date: 2021-01-07 22:43:44
  • Modify Date: 2024-01-03 10:50:45
  • (Pro3) GIP, human ((Pro3) Gastric Inhibitory Peptide, human) is an efficacious, stable and specific human GIP receptor (hGIPR) full agonist. (Pro3) GIP, human has high binding affinity for human GIPR with Ki/ Kd values of 0.90 nM. (Pro3) GIP, human can be used for the research of obesity-related diabetes[1][2].

Name (Pro3)-Gastric Inhibitory Polypeptide (human) trifluoroacetate salt
Description (Pro3) GIP, human ((Pro3) Gastric Inhibitory Peptide, human) is an efficacious, stable and specific human GIP receptor (hGIPR) full agonist. (Pro3) GIP, human has high binding affinity for human GIPR with Ki/ Kd values of 0.90 nM. (Pro3) GIP, human can be used for the research of obesity-related diabetes[1][2].
Related Catalog
Target

EC50: 0.026 nM (hGIPR)[2] Ki/Kd: 0.90 nM (hGIPR); 1.1 nM (Rat GIPR); 0.72 nM (Mouse GIPR)[2]

In Vitro (Pro3) GIP, human induces cAMP accumulation with an EC50 value of 0.026 nM[2]. (Pro3) GIP, human has high binding affinity for human GIPR, Rat GIPR and Mouse GIPR with Ki/ Kd values of 0.90 nM, 1.1 nM and 0.72 nM, respectively[2].
In Vivo (Pro3) GIP, human has comparatively weak partial agonist effect in rodent models[2].
Molecular Formula C226H338N60O64S