2304416-91-7

2304416-91-7 structure

Name: CBP/P300 bromodomain inhibitor-3
Chemical Name: CBP/P300 bromodomain inhibitor-3
CAS Number: 2304416-91-7
Molecular Formula: C₂₇H₃₁N₃O₄
Molecular Weight: 461.55
Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
Create Date: 2021-01-06 20:47:16
Modify Date: 2024-01-17 18:24:35
CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µΜ) and BRD4 (IC50=1-1000 µΜ) activity[1].

Name	CBP/P300 bromodomain inhibitor-3

Description	CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µΜ) and BRD4 (IC50=1-1000 µΜ) activity[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
Target	BRD4:1-1000 μM (IC50) CBP:0.01-0.1 μM (IC50)
References	[1]. Shawn E.R. Schiller, et al. Tetrahydro-imidazo quinoline compositions as cbp/p300 inhibitors. WO2019055877A1.

Molecular Formula	C₂₇H₃₁N₃O₄
Molecular Weight	461.55