CBP/P300 bromodomain inhibitor-3

Modify Date: 2024-01-17 18:24:35

CBP/P300 bromodomain inhibitor-3 Structure
CBP/P300 bromodomain inhibitor-3 structure
Common Name CBP/P300 bromodomain inhibitor-3
CAS Number 2304416-91-7 Molecular Weight 461.55
Density N/A Boiling Point N/A
Molecular Formula C27H31N3O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CBP/P300 bromodomain inhibitor-3


CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µΜ) and BRD4 (IC50=1-1000 µΜ) activity[1].

 Names

Name CBP/P300 bromodomain inhibitor-3

 CBP/P300 bromodomain inhibitor-3 Biological Activity

Description CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µΜ) and BRD4 (IC50=1-1000 µΜ) activity[1].
Related Catalog
Target

BRD4:1-1000 μM (IC50)

CBP:0.01-0.1 μM (IC50)

References

[1]. Shawn E.R. Schiller, et al. Tetrahydro-imidazo quinoline compositions as cbp/p300 inhibitors. WO2019055877A1.

 Chemical & Physical Properties

Molecular Formula C27H31N3O4
Molecular Weight 461.55