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2697176-16-0

2697176-16-0 structure
2697176-16-0 structure
  • Name: EPZ-719
  • Chemical Name: EPZ-719
  • CAS Number: 2697176-16-0
  • Molecular Formula: C22H31FN4O3S
  • Molecular Weight: 450.57
  • Catalog: Signaling Pathways Epigenetics Histone Methyltransferase
  • Create Date: 2022-01-07 19:14:08
  • Modify Date: 2024-01-09 12:59:52
  • EPZ-719 is a novel and potent SETD2 inhibitor ( IC50 = 0.005 μM) with a high selectivity over other histone methyltransferases.

Name EPZ-719
Description EPZ-719 is a novel and potent SETD2 inhibitor ( IC50 = 0.005 μM) with a high selectivity over other histone methyltransferases.
Related Catalog
References

[1]. Lampe JW, et al. Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical Studies. ACS Med Chem Lett. 2021 Aug 24;12(10):1539-1545.

Molecular Formula C22H31FN4O3S
Molecular Weight 450.57