2250132-99-9
2250132-99-9 structure
- Name: JTP-117968
- Chemical Name: JTP-117968
- CAS Number: 2250132-99-9
- Molecular Formula: C31H31F3N2O2
- Molecular Weight: 520.59
- Catalog: Signaling Pathways GPCR/G Protein Glucocorticoid Receptor
- Create Date: 2022-05-30 19:01:17
- Modify Date: 2024-01-14 09:36:18
-
JTP-117968, a novel selective glucocorticoid receptor modulator (a non-steroidal SGRM, IC50 of 6.8 nM), exhibits improved transrepression/transactivation dissociation[1].
| Name | JTP-117968 |
|---|
| Description | JTP-117968, a novel selective glucocorticoid receptor modulator (a non-steroidal SGRM, IC50 of 6.8 nM), exhibits improved transrepression/transactivation dissociation[1]. |
|---|---|
| Related Catalog | |
| In Vitro | JTP-117968 has partial TR activity, but exhibits extremely low TA activity[1]. |
| References |
| Molecular Formula | C31H31F3N2O2 |
|---|---|
| Molecular Weight | 520.59 |