2304852-21-7
2304852-21-7 structure
- Name: PAD-IN-2
- Chemical Name: PAD-IN-2
- CAS Number: 2304852-21-7
- Molecular Formula: C27H28ClN5O2
- Molecular Weight: 490.00
- Catalog: Research Areas Cancer
- Create Date: 2022-10-12 06:53:31
- Modify Date: 2024-09-24 10:58:33
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PAD-IN-2 is a potent pad4 inhibitor (IC50: <1 μM). PAD-IN-2 can be used in the research of auto-immune diseases and cancers, such as rheumatoid arthritis, vasculitis, systemic lupus erythematosis, cutaneous lupus erythematosis, ulcerative colitis, cystic fibrosis, asthma, multiple sclerosis and psoriasis[1].
| Name | PAD-IN-2 |
|---|
| Description | PAD-IN-2 is a potent pad4 inhibitor (IC50: <1 μM). PAD-IN-2 can be used in the research of auto-immune diseases and cancers, such as rheumatoid arthritis, vasculitis, systemic lupus erythematosis, cutaneous lupus erythematosis, ulcerative colitis, cystic fibrosis, asthma, multiple sclerosis and psoriasis[1]. |
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| Related Catalog | |
| In Vitro | PAD-IN-2 (Example-57, 1 h) inhibits PAD4 activity with an IC50 value <1 μM (determined by ammonia release biochemical assay)[1]. |
| References |
[1]. Hallur, Gurulingappa, et al. Heterocyclic compounds as pad4 inhibitors. Patent WO2019058393 A1. |
| Molecular Formula | C27H28ClN5O2 |
|---|---|
| Molecular Weight | 490.00 |