Shanghai Nianxing Industrial Co., Ltd
China
Product Name: Gsk466317a
Price: Check
Purity: 98.0%
Stocking Period: 10 Day
Contact: Yang
Email: sales@echemcloud.com

DC Chemicals Limited
China
Product Name: Gsk466317a
Price: ￥Inquiry/100mg ￥Inquiry/250mg ￥Inquiry/1g
Purity: 98.0%
Stocking Period: 10 Day
Contact: Tony Cao
Email: sales@dcchemicals.com

864082-48-4

864082-48-4 structure

864082-48-4 structure

Name: Gsk466317a
Chemical Name: GSK466317A
CAS Number: 864082-48-4
Molecular Formula: C₂₁H₁₆ClF₃N₄O₂
Molecular Weight: 448.83
Catalog: Signaling Pathways Protein Tyrosine Kinase/RTK PKA
Create Date: 2023-09-26 13:02:57
Modify Date: 2024-01-16 11:39:22
GSK466317A is a PKA inhibitor, with an IC50 of 12.59 μM. GSK466317A also inhibits GRK1, GRK2, and GRK5, with IC50s of 1000, 31.62, and 39.81 μM, respectively[1].

Name	GSK466317A

Description	GSK466317A is a PKA inhibitor, with an IC50 of 12.59 μM. GSK466317A also inhibits GRK1, GRK2, and GRK5, with IC50s of 1000, 31.62, and 39.81 μM, respectively[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Protein Tyrosine Kinase/RTK >> PKA Signaling Pathways >> Stem Cell/Wnt >> PKA Research Areas >> Neurological Disease
Target	PKA:12.59 μM (IC50)
References	[1]. Homan KT, et, al. Identification and structure-function analysis of subfamily selective G protein-coupled receptor kinase inhibitors. ACS Chem Biol. 2015 Jan 16;10(1):310-9.

Molecular Formula	C₂₁H₁₆ClF₃N₄O₂
Molecular Weight	448.83

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