- Shanghai Nianxing Industrial Co., Ltd
- China
- Product Name: Varenicline Tartrate
- Price:
- Purity: 98.0%
- Stocking Period: 10 Day
- Contact: Yang
- Shanghai Jizhi Biochemical Technology Co., Ltd
- China
- Product Name: Varenicline Tartrate
- Price: ￥2108.0/25mg ￥1058.0/5mg ￥688.0/20mg
- Purity: 98.0%
- Stocking Period: Inquiry
- Contact: Liu jia
- ShangHai DC Chemicals Co.,Ltd
- China
- Product Name: Varenicline tartrate
- Price: ￥Inquiry/1g
- Purity: 98.9%
- Stocking Period: 1 Day
- Contact: Tony Lai
- DC Chemicals Limited
- China
- Product Name: Varenicline tartrate
- Price: $200.0/100mg $400.0/250mg $800.0/1g
- Purity: 98.0%
- Stocking Period: 3 Day
- Contact: Tony Cao
- Dayang Chem (Hangzhou) Co., Ltd.
- China
- Product Name: Varenicline tartrate
- Price: $Inquiry/100g $Inquiry/1kg $Inquiry/100kg $Inquiry/1000kg
- Purity: 98.0%
- Stocking Period: Inquiry
- Contact: Ms Wang
375815-87-5
375815-87-5 structure
- Name: Varenicline Tartrate
- Chemical Name: varenicline tartrate
- CAS Number: 375815-87-5
- Molecular Formula: C17H19N3O6
- Molecular Weight: 361.35
- Catalog: Biochemical Inhibitor Neuronal Signaling AChR agonist
- Create Date: 2018-06-20 23:03:29
- Modify Date: 2024-01-02 18:18:16
-
Varenicline Tartrate(CP 526555;Champix) is a nicotinic receptor partial agonist; it stimulates nicotine receptors more weakly than nicotine itself does.IC50 value:Target: α4β2 nAChRVarenicline(CP 526555; Champix; Chantix) is a prescription medication used to treat smoking addiction. As a partial agonist it both reduces cravings for and decreases the pleasurable effects of cigarettes and other tobacco products. Through these mechanisms Varenicline(CP 526555; Champix; Chantix) can assist some patients to quit smoking.
| Name | varenicline tartrate |
|---|---|
| Synonyms |
7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine tartrate Champix
(2R,3R)-3-carboxy-2,3-dihydroxypropanoate de (1R,12S)-5,8-diaza-14-azoniatétracyclo[10.3.1.0.0]hexadéca-2(11),3,5,7,9-pentaène Chantix (1R,12S)-5,8-Diaza-14-azoniatetracyclo[10.3.1.0.0]hexadeca-2(11),3,5,7,9-pentaene (2R,3R)-3-carboxy-2,3-dihydroxypropanoate (1R,12S)-5,8-Diaza-14-azoniatetracyclo[10.3.1.0.0]hexadeca-2(11),3,5,7,9-pentaen-(2R,3R)-3-carboxy-2,3-dihydroxypropanoat Butanedioic acid, 2,3-dihydroxy-, (2R,3R)-, compd. with (6R,10S)-7,8,9,10-tetrahydro-6,10-methano-6H-azepino[4,5-g]quinoxaline (1:1) Champix Varenicline tartrate |
| Description | Varenicline Tartrate(CP 526555;Champix) is a nicotinic receptor partial agonist; it stimulates nicotine receptors more weakly than nicotine itself does.IC50 value:Target: α4β2 nAChRVarenicline(CP 526555; Champix; Chantix) is a prescription medication used to treat smoking addiction. As a partial agonist it both reduces cravings for and decreases the pleasurable effects of cigarettes and other tobacco products. Through these mechanisms Varenicline(CP 526555; Champix; Chantix) can assist some patients to quit smoking. |
|---|---|
| Related Catalog | |
| References |
[5]. Varenicline |
| Boiling Point | 400.6ºC at 760 mmHg |
|---|---|
| Melting Point | 206-208ºC |
| Molecular Formula | C17H19N3O6 |
| Molecular Weight | 361.35 |
| PSA | 23.79000 |
| LogP | 4.49528 |
| Storage condition | Desiccate at RT |
| Water Solubility | DMSO: >5mg/mL |
| Symbol |
GHS02, GHS06, GHS08 |
|---|---|
| Signal Word | Danger |
| Hazard Statements | H225-H301 + H311 + H331-H370 |
| Precautionary Statements | P210-P260-P280-P301 + P310-P311 |
| Hazard Codes | Xn,N,T,F |
| Risk Phrases | 22-50-39/23/24/25-23/24/25-11 |
| Safety Phrases | 22-57-45-36/37-16-7 |
| RIDADR | UN 3077 9 / PGIII |
| Flash Point(F) | 48.2 °F |
| Flash Point(C) | 9 °C |
|
~64%
375815-87-5 |
| Literature: Medichem, S.A. Patent: US2012/4239 A1, 2012 ; Location in patent: Page/Page column 12 ; |
| Precursor 2 | |
|---|---|
| DownStream 0 | |