63-12-7

63-12-7 structure

Name: benzquinamide
Chemical Name: benzquinamide
CAS Number: 63-12-7
Molecular Formula: C₂₂H₃₂N₂O₅
Molecular Weight: 404.50000
Catalog: Signaling Pathways GPCR/G Protein Adrenergic Receptor
Create Date: 2017-06-13 06:05:05
Modify Date: 2024-01-13 12:57:24
Benzquinamide is an antiemetic which can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) with Ki values of 1,365, 691, and 545 nM, respectively.

Name	benzquinamide
Synonyms	P2647

Description	Benzquinamide is an antiemetic which can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) with Ki values of 1,365, 691, and 545 nM, respectively.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Adrenergic Receptor Research Areas >> Metabolic Disease
Target	Ki: 1,365 nM (α2A), 691 nM (α2B), 545 nM (α2C)[1].
References	[1]. Elisabet Gregori-Puigjané, et al. Identifying mechanism-of-action targets for drugs and probes. Proc Natl Acad Sci U S A. 2012 Jul 10; 109(28): 11178-11183. doi: 10.1073/pnas.1204524109