BRL 52537 HYDROCHLORIDE structure
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Common Name | BRL 52537 HYDROCHLORIDE | ||
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CAS Number | 112282-24-3 | Molecular Weight | 391.76 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C18H25Cl3N2O | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of BRL 52537 HYDROCHLORIDEBRL 52537 hydrochloride is a highly selective κ-Opioid receptor (KOR) agonist with Kis of 0.24 nM and 1560 nM for κ and μ subtypes, respectively. BRL 52537 hydrochloride decreases ischemia-evoked NO production as a potential mechanism of neuroprotection. BRL 52537 hydrochloride attenuates early stroke damage[1]. |
Name | BRL 52537 hydrochloride |
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Synonym | More Synonyms |
Description | BRL 52537 hydrochloride is a highly selective κ-Opioid receptor (KOR) agonist with Kis of 0.24 nM and 1560 nM for κ and μ subtypes, respectively. BRL 52537 hydrochloride decreases ischemia-evoked NO production as a potential mechanism of neuroprotection. BRL 52537 hydrochloride attenuates early stroke damage[1]. |
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Related Catalog | |
Target |
Ki: 0.24 nM (κ-Opioid receptor) and 1560 nM (μ-Opioid receptor)[1] |
References |
Molecular Formula | C18H25Cl3N2O |
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Molecular Weight | 391.76 |
Exact Mass | 390.103241 |
PSA | 23.55000 |
LogP | 4.69060 |
Storage condition | 2-8°C |
Hazard Codes | Xi |
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