BMS-986163 structure
|
Common Name | BMS-986163 | ||
|---|---|---|---|---|
| CAS Number | 1801151-09-6 | Molecular Weight | 462.45 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C23H28FN2O5P | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of BMS-986163BMS-986163 is a negative allosteric modulator of GluN2B. The prodrug BMS-986163 rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM). |
| Name | BMS-986163 |
|---|
| Description | BMS-986163 is a negative allosteric modulator of GluN2B. The prodrug BMS-986163 rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM). |
|---|---|
| Related Catalog | |
| Target |
IC50: 4 nM (GluN2B, BMS-986169), 24 nM (GluN2B, BMS-986169)[1] |
| References |
| Molecular Formula | C23H28FN2O5P |
|---|---|
| Molecular Weight | 462.45 |
| InChIKey | ZPUVTBAQHJFPHE-BHDDXSALSA-N |
| SMILES | Cc1ccc(CN2CCC(N3CCC(c4ccc(OP(=O)(O)O)cc4)C(F)C3)C2=O)cc1 |