DKFZ-251

Modify Date: 2023-10-16 13:36:37

DKFZ-251 Structure
DKFZ-251 structure
Common Name DKFZ-251
CAS Number 2222059-70-1 Molecular Weight 416.481
Density N/A Boiling Point N/A
Molecular Formula C24H24N4O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of DKFZ-251


DKFZ-251 (DKFZ251) is a selective inhibitor of Kallikrein-related peptidase 6 (KLK6) with IC50 of 0.13 uM, demonstrates good selectivity for KLK6 compared to other KLKs; DKFZ-633 exhibits on-target activity in a cellular assay.

 Names

Name DKFZ-251

 DKFZ-251 Biological Activity

Description DKFZ-251 (DKFZ251) is a selective inhibitor of Kallikrein-related peptidase 6 (KLK6) with IC50 of 0.13 uM, demonstrates good selectivity for KLK6 compared to other KLKs; DKFZ-633 exhibits on-target activity in a cellular assay.
References References 1. De Vita E, et al. J Med Chem. 2018 Sep 28. doi: 10.1021/acs.jmedchem.8b01106. View Related Products by Target Other Targets

 Chemical & Physical Properties

Molecular Formula C24H24N4O3
Molecular Weight 416.481