PROTAC MEK1 Degrader-1

Modify Date: 2025-10-03 11:54:19

PROTAC MEK1 Degrader-1 Structure
PROTAC MEK1 Degrader-1 structure
 Common Name PROTAC MEK1 Degrader-1
CAS Number 2671004-41-2 Molecular Weight 1201.17
Density N/A Boiling Point N/A
Molecular Formula C53H66FIN8O11S2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of PROTAC MEK1 Degrader-1


PROTAC MEK1 Degrader-1 is a PROTAC targeting MEK1 with a pIC50 value of 7.0. PROTAC MEK1 Degrader-1 consists of a MEK1 inhibitor and a von Hippel-Lindau ligand. PROTAC MEK1 Degrader-1 can inhibit ERK1/2 phosphorylation. PROTAC MEK1 Degrader-1 shows an antiproliferative activity against A375 cells[1].

 Names

Name PROTAC MEK1 Degrader-1

 PROTAC MEK1 Degrader-1 Biological Activity

Description PROTAC MEK1 Degrader-1 is a PROTAC targeting MEK1 with a pIC50 value of 7.0. PROTAC MEK1 Degrader-1 consists of a MEK1 inhibitor and a von Hippel-Lindau ligand. PROTAC MEK1 Degrader-1 can inhibit ERK1/2 phosphorylation. PROTAC MEK1 Degrader-1 shows an antiproliferative activity against A375 cells[1].
Related Catalog
References

[1]. Vollmer S, et al. Design, Synthesis, and Biological Evaluation of MEK PROTACs. J Med Chem. 2020 Jan 9;63(1):157-162.  

 Chemical & Physical Properties

Molecular Formula C53H66FIN8O11S2
Molecular Weight 1201.17
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Chemsrc provides PROTAC MEK1 Degrader-1(CAS#:2671004-41-2) MSDS, density, melting point, boiling point, structure, formula, molecular weight etc. Articles of PROTAC MEK1 Degrader-1 are included as well.>> amp version: PROTAC MEK1 Degrader-1

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