LUF 5834
Modify Date: 2025-08-25 16:56:38
LUF 5834 structure
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Common Name | LUF 5834 | ||
|---|---|---|---|---|
| CAS Number | 333962-91-7 | Molecular Weight | 348.38 | |
| Density | 1.5±0.1 g/cm3 | Boiling Point | 655.8±65.0 °C at 760 mmHg | |
| Molecular Formula | C17H12N6OS | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 350.4±34.3 °C | |
Use of LUF 5834LUF5834 is a selective A2B adenosine receptor (A2BR) partial agonist (EC50 = 12 nM). LUF5834 is also a partial A1/A2A adenosine receptor agonist (lacking selectivity) with Ki values of 2.6 and 28 nM, respectively[1][2]. |
| Name | LUF5834 |
|---|---|
| Synonym | More Synonyms |
| Description | LUF5834 is a selective A2B adenosine receptor (A2BR) partial agonist (EC50 = 12 nM). LUF5834 is also a partial A1/A2A adenosine receptor agonist (lacking selectivity) with Ki values of 2.6 and 28 nM, respectively[1][2]. |
|---|---|
| Related Catalog | |
| Target |
A2BR:12 nM (EC50) A2AR:28 nM (Ki) A1R:2.6 nM (Ki) |
| References |
| Density | 1.5±0.1 g/cm3 |
|---|---|
| Boiling Point | 655.8±65.0 °C at 760 mmHg |
| Molecular Formula | C17H12N6OS |
| Molecular Weight | 348.38 |
| Flash Point | 350.4±34.3 °C |
| Exact Mass | 348.079315 |
| LogP | 2.75 |
| Vapour Pressure | 0.0±2.0 mmHg at 25°C |
| Index of Refraction | 1.753 |
| 2-Amino-4-(4-hydroxyphenyl)-6-[(2H-imidazol-2-ylmethyl)sulfanyl]-3,5-pyridinedicarbonitrile |
| 3,5-Pyridinedicarbonitrile, 2-amino-4-(4-hydroxyphenyl)-6-[(2H-imidazol-2-ylmethyl)thio]- |
| LUF5834 |
| 2-amino-4-(4-hydroxyphenyl)-6-(1H-imidazol-2-ylmethylsulfanyl)pyridine-3,5-dicarbonitrile |