Meptazinol HCl
Meptazinol HCl structure
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Common Name | Meptazinol HCl | ||
|---|---|---|---|---|
| CAS Number | 59263-76-2 | Molecular Weight | 269.810 | |
| Density | N/A | Boiling Point | 354.8ºC at 760 mmHg | |
| Molecular Formula | C15H24ClNO | Melting Point | 250-252ºC | |
| MSDS | Chinese USA | Flash Point | 160.6ºC | |
| Symbol |
GHS07 |
Signal Word | Warning | |
Use of Meptazinol HClMeptazinol Hcl(WY-22811 Hcl) is a unique centrally active opioid analgesic. |
| Name | Meptazinol Hydrochloride |
|---|---|
| Synonym | More Synonyms |
| Boiling Point | 354.8ºC at 760 mmHg |
|---|---|
| Melting Point | 250-252ºC |
| Molecular Formula | C15H24ClNO |
| Molecular Weight | 269.810 |
| Flash Point | 160.6ºC |
| Exact Mass | 269.154633 |
| PSA | 23.47000 |
| LogP | 3.89560 |
| InChIKey | MPJUSISYVXABBH-UHFFFAOYSA-N |
| SMILES | CCC1(c2cccc(O)c2)CCCCN(C)C1.Cl |
| Storage condition | Desiccate at +4°C |
| Water Solubility | H2O: >10mg/mL |
CHEMICAL IDENTIFICATION
HEALTH HAZARD DATAACUTE TOXICITY DATA
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~91%
Meptazinol HCl CAS#:59263-76-2 |
| Literature: Bradley; Cavalla; Edington; et al. European Journal of Medicinal Chemistry, 1980 , vol. 15, # 4 p. 375 - 385 |
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Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
|
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Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
|
~%
Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
|
~%
Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
|
~%
Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
|
~%
Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
|
~%
Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
|
~%
Meptazinol HCl CAS#:59263-76-2 |
| Literature: European Journal of Medicinal Chemistry, , vol. 15, # 4 p. 375 - 385 |
| Precursor 10 | |
|---|---|
| DownStream 1 | |
CAS#:54340-58-8| HS Code | 2942000000 |
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Bis(9)-(-)-nor-meptazinol as a novel dual-binding AChEI potently ameliorates scopolamine-induced cognitive deficits in mice.
Pharmacol. Biochem. Behav. 104 , 138-43, (2013) Alzheimer's disease (AD) is a multifaceted neurodegenerative disorder which is characterized by the progressive deterioration of cognition and the emergence of behavioral and psychological symptoms in... |
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Reflex activity caused by laryngoscopy and intubation is obtunded differently by meptazinol, nalbuphine and fentanyl.
Eur. J. Anaesthesiol. 24(1) , 53-8, (2007) To evaluate the different potencies of several opioids in obtunding reflex mechanisms of laryngoscopy and intubation.Three groups of patients (each n = 25, ASA 1-2) undergoing elective plastic surgery... |
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Lack of sensitization during place conditioning in rats is consistent with the low abuse potential of tramadol.
Neurosci. Lett. 329(1) , 25-8, (2002) Based on the recent finding that tramadol (TRAM) produces conditioned place preference (CPP) and dopamine release in the nucleus accumbens, it was suggested that the abuse liability of TRAM may be gre... |
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Name: Luminescence-based cell-based primary high throughput screening assay to identify ago...
Source: The Scripps Research Institute Molecular Screening Center
Target: mu-type opioid receptor isoform MOR-1 [Homo sapiens]
External Id: OPRM1-OPRD1_AG_LUMI_1536_1X%ACT PRUN
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Name: Primary qHTS assay for inhibitors of alpha-synuclein gene (SNCA) expression
Source: NCGC
External Id: SNCA-p-activity-luciferase
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Name: Fluorescence-based cell-based primary high throughput screening assay to identify ago...
Source: The Scripps Research Institute Molecular Screening Center
Target: muscarinic acetylcholine receptor M1 [Homo sapiens]
External Id: CHRM1_AG_FLUO8_1536_1X%ACT PRUN
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Name: Cytochrome P450 Family 1 Subfamily A Member 2 (CYP1A2) small molecule antagonists: lu...
Source: 824
External Id: CYP273
|
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Name: Dicer-mediated maturation of pre-microRNA
Source: Center for Chemical Genomics, University of Michigan
Target: N/A
External Id: TargetID_659_CEMA
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|
Name: Fluorescence-based cell-based primary high throughput screening assay to identify pos...
Source: The Scripps Research Institute Molecular Screening Center
Target: muscarinic acetylcholine receptor M1 [Homo sapiens]
External Id: CHRM1_PAM_FLUO8_1536_1X%ACT PRUN
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|
Name: Fluorescence polarization-based biochemical high throughput primary assay to identify...
Source: The Scripps Research Institute Molecular Screening Center
Target: RecName: Full=Sialate O-acetylesterase; AltName: Full=H-Lse; AltName: Full=Sialic acid-specific 9-O-acetylesterase; Flags: Precursor [Homo sapiens]
External Id: SIAE_INH_FP_1536_1X%INH PRUN
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Name: p53 small molecule agonists, cell-based qHTS assay: qHTS cell viability counter scree...
Source: 824
Target: N/A
External Id: P53600
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Name: p53 small molecule agonists, cell-based qHTS assay with rat liver microsomes: qHTS ce...
Source: 824
Target: N/A
External Id: P53MS958
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Name: p53 small molecule agonists, cell-based qHTS assay with rat liver microsomes: Summary
Source: 824
External Id: P53MS482
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| Phenol, 3-(3-ethylhexahydro-1-methyl-1H-azepin-3-yl)-, hydrochloride (1:1) |
| 3-(3-Ethyl-1-methylazepan-3-yl)phenol hydrochloride (1:1) |
| 3-(3-ethyl-1-methylazepan-3-yl)phenol,hydrochloride |
| 3-(3-Ethyl-1-methyl-3-azepanyl)phenol hydrochloride (1:1) |
| UNII:T62FQ4ZCPA |
| MEPTAZINOL HYDROCHLORIDE |