Cicloprolol hydrochloride

Modify Date: 2024-01-03 18:07:30

Cicloprolol hydrochloride Structure
Cicloprolol hydrochloride structure
Common Name Cicloprolol hydrochloride
CAS Number 63686-79-3 Molecular Weight 359.888
Density N/A Boiling Point N/A
Molecular Formula C18H30ClNO4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Cicloprolol hydrochloride


Cicloprolol is a partial β 1-adrenoceptor agonist .

 Names

Name Cicloprolol hydrochloride
Synonym More Synonyms

 Cicloprolol hydrochloride Biological Activity

Description Cicloprolol is a partial β 1-adrenoceptor agonist .
Related Catalog
Target

Adrenoceptor[1]

In Vitro Cicloprolol is a partial β1-adrenoceptor agonist considered for the treatment of patients with coronary artery disease and impaired left ventricular function[1]. The new β-adrenoceptor partial agonist Cicloprolol acts as a β-agonist at normal levels and as a β-antagonist at high levels of adrenergic discharge. Treatment with Cicloprolol should protect the heart against excessive stimulation, while providing a baseline level of sympathetic drive. Cicloprolol has a weak β1-agonistic effect at normal levels of adrenergic discharge and acts as an antagonist at high levels of discharge[2].
References

[1]. Weber S, et al. Pharmacodynamic without pharmacokinetic interaction between cicloprolol, a partial beta 1-adrenoceptor agonist, and digoxin in healthy subjects. Br J Clin Pharmacol. 1990 Sep;30(3):411-6

[2]. Cocco G, et al. An evaluation of the safety of the beta-modulator cicloprolol in chronic heart failure. Clin Cardiol. 1992 Jan;15(1):38-42.

 Chemical & Physical Properties

Molecular Formula C18H30ClNO4
Molecular Weight 359.888
Exact Mass 359.186340

 Synonyms

(±)-1-(p-(2-(Cyclopropylmethoxy)ethoxy)phenoxy)-3-(isopropylamino)-2-propanol Hydrochloride
1-{4-[2-(Cyclopropylmethoxy)ethoxy]phenoxy}-3-(isopropylamino)-2-propanol hydrochloride (1:1)
2-Propanol, 1-[4-[2-(cyclopropylmethoxy)ethoxy]phenoxy]-3-[(1-methylethyl)amino]-, hydrochloride (1:1)
(±)-1-(4-(2-(Cyclopropylmethoxy)ethoxy)phenoxy)-3-((1-methylethyl)amino)-2-propanol Hydrochloride
cicloprolol hydrochloride
sl-d 177
UNII:T355YD4791
T355YD4791
Top Suppliers:I want be here


Get all suppliers and price by the below link:

Cicloprolol hydrochloride suppliers


Price: $696/1mg

Reference only. check more Cicloprolol hydrochloride price