Setastine

Modify Date: 2024-01-05 18:20:40

Setastine Structure
Setastine structure
Common Name Setastine
CAS Number 64294-95-7 Molecular Weight 357.91700
Density N/A Boiling Point N/A
Molecular Formula C22H28ClNO Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Setastine


Setastine (EGIS-2062 (free acid); EGYT-2062 (free acid) is an orally effective, non-sedative and long acting anti-allergic agent. Setastine possesses potent histamine Hi-receptor blocking properties and can be used for allergies and rhinitis research[1]<.

 Names

Name 1-[2-[1-(4-chlorophenyl)-1-phenylethoxy]ethyl]azepane
Synonym More Synonyms

 Setastine Biological Activity

Description Setastine (EGIS-2062 (free acid); EGYT-2062 (free acid) is an orally effective, non-sedative and long acting anti-allergic agent. Setastine possesses potent histamine Hi-receptor blocking properties and can be used for allergies and rhinitis research[1]<.
Related Catalog
Target

IC50:Histamine Hi-receptor[1]

References

[1]. Németh, A., & Huszti, Z. (1988). The effect of a new antihistamine drug, Loderix® (EGIS-2062), on stimulus-evoked histamine release from rat peritoneal mast cells. Agents and Actions, 23(3-4), 194–197.  

 Chemical & Physical Properties

Molecular Formula C22H28ClNO
Molecular Weight 357.91700
Exact Mass 357.18600
PSA 12.47000
LogP 5.43400

 Safety Information

HS Code 2933990090

 Customs

HS Code 2933990090
Summary 2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

 Synonyms

1H-Azepine,1-(2-(1-(4-chlorophenyl)-1-phenylethoxy)ethyl)hexahydro
Setastine
Setastine [INN]
Setastina
Setastinum
1-(2-(1-(4-Chlorophenyl)-1-phenylethoxy)ethyl)azepane
Setastinum [INN-Latin]