CARM1-IN-3

Modify Date: 2024-01-17 23:29:58

CARM1-IN-3 Structure
CARM1-IN-3 structure
Common Name CARM1-IN-3
CAS Number 912970-67-3 Molecular Weight 408.54
Density N/A Boiling Point N/A
Molecular Formula C24H32N4O2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CARM1-IN-3


CARM1-IN-3 (compound 17b) is a potent and selective co-activator associated arginine methyltransferase (CARM1) inhibitor with IC50 values of 0.07, >25 µM for CARM1 and CARM3, respectively[1].

 Names

Name CARM1-IN-3

 CARM1-IN-3 Biological Activity

Description CARM1-IN-3 (compound 17b) is a potent and selective co-activator associated arginine methyltransferase (CARM1) inhibitor with IC50 values of 0.07, >25 µM for CARM1 and CARM3, respectively[1].
Related Catalog
Target

IC50: 0.07 µM (CARM1); >25 µM (CARM3)[1]

References

[1]. Wan H, et al. Benzo[d]imidazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1)--Hit to Lead studies. Bioorg Med Chem Lett. 2009 Sep 1;19(17):5063-6.  

 Chemical & Physical Properties

Molecular Formula C24H32N4O2
Molecular Weight 408.54
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.