麻醉椒苦素

Methylsticin 是从卡瓦根中分离出来的一种卡瓦内酯。Methylsticin 具有抑制破骨细胞形成的活性。

[ 描述 ]:

[ 相关类别 ]:

[参考文献]

[ 密度 ]:
1.3±0.1 g/cm3

[ 沸点 ]:
496.5±45.0 °C at 760 mmHg

[ 熔点 ]:
139-140.5ºC

[ 分子式 ]:
C₁₅H₁₄O₅

[ 分子量 ]:
274.269

[ 闪点 ]:
223.9±28.8 °C

[ 精确质量 ]:
274.084137

[ PSA ]:
53.99000

[ LogP ]:
1.81

[ 外观性状 ]:
白色粉末

[ 蒸汽压 ]:
0.0±1.3 mmHg at 25°C

[ 折射率 ]:
1.597

[ 储存条件 ]:
2-8°C

CHEMICAL IDENTIFICATION

RTECS NUMBER :

UQ0517000

CHEMICAL NAME :

2H-Pyran-2-one, 5,6-dihydro-4-methoxy-6-(3,4-(methylenedioxy)styryl)- , (R)-

CAS REGISTRY NUMBER :

495-85-2

BEILSTEIN REFERENCE NO. :

0091701

LAST UPDATED :

199612

DATA ITEMS CITED :

2

MOLECULAR FORMULA :

C15-H14-O5

MOLECULAR WEIGHT :

274.29

WISWESSER LINE NOTATION :

T56 BO DO CHJ G1U1- FT6OV CUTJ DO1

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :

LD50 - Lethal dose, 50 percent kill

ROUTE OF EXPOSURE :

Intraperitoneal

SPECIES OBSERVED :

Rodent - mouse

DOSE/DURATION :

530 mg/kg

TOXIC EFFECTS :

Behavioral - anticonvulsant

REFERENCE :

AIPTAK Archives Internationales de Pharmacodynamie et de Therapie. (Heymans Institute of Pharmacology, De Pintelaan 185, B-9000 Ghent, Belgium) V.4- 1898- Volume(issue)/page/year: 177,261,1969

TYPE OF TEST :

LD50 - Lethal dose, 50 percent kill

ROUTE OF EXPOSURE :

Intravenous

SPECIES OBSERVED :

Rodent - mouse

DOSE/DURATION :

49 mg/kg

TOXIC EFFECTS :

Behavioral - anticonvulsant

REFERENCE :

AIPTAK Archives Internationales de Pharmacodynamie et de Therapie. (Heymans Institute of Pharmacology, De Pintelaan 185, B-9000 Ghent, Belgium) V.4- 1898- Volume(issue)/page/year: 177,261,1969

[ 危险品运输编码 ]:
NONH for all modes of transport

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公司名：上海化源世纪贸易有限公司

区域：上海市普陀区

价格：

联系人：徐乾明

产品详情：麻醉椒苦素

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公司名：上海源溪生物科技有限公司

区域：上海市浦东新区

价格：
￥需询单/1g

联系人：赖经理

产品详情：Kavatin

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