纳曲吲哚盐酸盐

纳曲吲哚盐酸盐结构式
纳曲吲哚盐酸盐结构式
品牌特惠专场
常用名 纳曲吲哚盐酸盐 英文名 Naltrindole hydrochloride
CAS号 111469-81-9 分子量 450.95700
密度 N/A 沸点 664.2ºC at 760mmHg
分子式 C26H27ClN2O3 熔点 N/A
MSDS 中文版 美版 闪点 355.5ºC

Naltrindole, a highly selective and potent non-peptide delta opioid receptor antagonist.

Eur. J. Pharmacol. 146 , 185, (1988)

Acute delta-opioid receptor activation induces CREB phosphorylation in NG108-15 cells.

Eur. J. Pharmacol. 390 , 1-6, (2000)

A growing body of evidence supports an important role of the transcription factor cAMP responsive element binding protein (CREB) in mediating opioid-induced changes in the cAMP pathway. Regulation of CREB and subsequent changes in gene expression may underlie...

Characterization of delta-opioid receptors and effect of enkephalins on IRD 98 rat epithelial intestinal cell line.

Pflugers Arch. 439 , 547-554, (2000)

Using 3H-Tyr-D-Ala-Gly-Phe-D-Leu-OH (3H-DADLE) as a radioligand, delta-opioid binding sites on the IRD 98 rat epithelial cell line were identified. These sites were found to be reversible, saturable, specific and displayed high affinity for DADLE. Scatchard a...