| 常用名 | Ex26 | CAS号 | 1233332-37-0 |
|---|---|---|---|
| 价格 | ¥7740.0/50mg ¥需询单/1g ¥需询单/1g ¥需询单/1g | 纯度 | 98.0% |
| 备货期 | 1天 | 库存 | 现货 |
| 产品网页 | http://www.aladdin-e.com/zh_cn/E286856.html | ||
| 产品详情(用途,包装等)
用途: Ex26 (S1P1-IN-Ex26) is a potent and selective Sphingosine 1-phosphate receptor 1 (S1P1) antagonist (IC50=0.93 nM). Ex26 shows >3,000-fold selectivity for S1P1 over other Sphingosine 1-phosphate receptors. Ex26 can be used in experimental autoimmune encephalomyelitis reseach[1]. 作用: 有力和选择性的S1P1受体拮抗剂(IC50 = 0.93 nM)。与S1P2,S1P3,S1P4和S1P5相比,S1P1的选择性> 3,000倍。在外周淋巴结中诱导淋巴细胞隔离并上调S1P1受体表达。降低EAE小鼠的疾病严重程度。增加体内刺激树突状细胞中IFN-α的产生。 物理化学性质: CAS号:1233332-37-0 常用中文名:Ex26 常用英文名:Ex26 分子式:C28H28ClFN2O3 分子量:494.98 密度:1.3±0.1 g/cm3 沸点:634.3±55.0 °C at 760 mmHg 熔点:N/A 闪点:337.4±31.5 °C 储存条件:2-8°C储存 |