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PROTAC CDK9 Degrader-1

更新时间:2025-08-27 07:59:35

PROTAC CDK9 Degrader-1结构式
PROTAC CDK9 Degrader-1结构式
品牌特惠专场
常用名 PROTAC CDK9 Degrader-1 英文名 PROTAC 6
CAS号 2118356-96-8 分子量 613.66
密度 N/A 沸点 N/A
分子式 C33H35N5O7 熔点 N/A
MSDS N/A 闪点 N/A

 PROTAC CDK9 Degrader-1用途


PROTAC 6 是一种有选择性的 CDK9 降解剂。

 PROTAC CDK9 Degrader-1名称

中文名 PROTAC CDK9 Degrader-1
英文名 PROTAC 6

 PROTAC CDK9 Degrader-1生物活性

描述 PROTAC CDK9 Degrader-1 是一种有选择性的 CDK9 降解剂。
相关类别
靶点实验

CDK9

参考文献

[1]. Robb CM, et al. Chemically induced degradation of CDK9 by a proteolysis targeting chimera (PROTAC). Chem Commun (Camb). 2017 Jul 4;53(54):7577-7580.

 PROTAC CDK9 Degrader-1物理化学性质

分子式 C33H35N5O7
分子量 613.66
储存条件 -20°C,密闭,干燥

 PROTAC CDK9 Degrader-1靶点实验

查看更多实验

实验名称:Protac activity at CRBN/CDK9 in human HCT116 cells assessed as induction of CDK9 prot...
来源:ChEMBL
靶标:Protein cereblon
External Id:CHEMBL4388616
实验名称:Protac activity at CRBN/CDK9 in human HCT-116 cells assessed as induction of CDK9 deg...
来源:ChEMBL
靶标:Protein cereblon
External Id:CHEMBL5230793
实验名称:Protac activity at CRBN/CDK9 in human HCT-116 cells assessed as induction of CDK9 deg...
来源:ChEMBL
靶标:Protein cereblon
External Id:CHEMBL5230794
实验名称:PROTAC activity at E3 ubiquitin ligase/CDK9 in human HCT-116 cells assessed as induct...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL5621183
实验名称:Protac activity at CRBN/CDK9 in human HCT-116 cells at 20 uM relative to control
来源:ChEMBL
靶标:Protein cereblon
External Id:CHEMBL5242525
实验名称:PROTAC activity at CRBN/CDK9 in human MV4-11 cells assessed as maximal degradation of...
来源:ChEMBL
靶标:Protein cereblon
External Id:CHEMBL5546630
实验名称:PROTAC activity at CRBN/CDK9 in human MV4-11 cells assessed as maximal degradation of...
来源:ChEMBL
靶标:Protein cereblon
External Id:CHEMBL5546631
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