杜鹃黄素

• 常用名: 杜鹃黄素
• 英文名: Azaleatin
• CAS号: 529-51-1
• 分子量: 316.26200
• 密度: 1.634g/cm3
• 沸点: 657.3ºC at 760mmHg
• 分子式: C₁₆H₁₂O₇
• 熔点: N/A
• 闪点: 250.2ºC

杜鹃黄素用途

Azaleatin 是一种从 Rhododendron 种中分离得到的 O-甲基化黄酮醇。Azaleatin 是二肽基肽酶-IV 的抑制剂。Azaleatin 可用于 2 型糖尿病和肥胖症的研究。

杜鹃黄素名称

• 中文名: 杜鹃黄素
• 英文名: azaleatin
• 中文别名: 2-(3,4-二羟基苯基)-3,7-二羟基-5-甲氧基苯并吡喃-4-酮

杜鹃黄素生物活性

• 描述: Azaleatin 是一种从 Rhododendron 种中分离得到的 O-甲基化黄酮醇。Azaleatin 是二肽基肽酶-IV 的抑制剂。Azaleatin 可用于 2 型糖尿病和肥胖症的研究。
• 相关类别:
  信号通路 >> 代谢酶/蛋白酶 >> 二肽基肽酶
  研究领域 >> 代谢疾病
• 靶点实验:

  Dipeptidyl Peptidase-IV Inhibitor[2]

• 参考文献:

  [1]. Harborne JB, et, al. Leaf survey of flavonoids and simple phenols in the genus Rhododendron. Phytochemistry. 1971 Nov; 10(11): 2727-2744.

  [2]. The medicinal usage of azaleatin. CN107375268A.

杜鹃黄素物理化学性质

• 密度: 1.634g/cm3
• 沸点: 657.3ºC at 760mmHg
• 分子式: C₁₆H₁₂O₇
• 分子量: 316.26200
• 闪点: 250.2ºC
• 精确质量: 316.05800
• PSA: 120.36000
• LogP: 2.29100
• InChIKey: RJBAXROZAXAEEM-UHFFFAOYSA-N
• SMILES: COc1cc(O)cc2oc(-c3ccc(O)c(O)c3)c(O)c(=O)c12
• 折射率: 1.74
• 储存条件: 2-8°C，密封，干燥

杜鹃黄素安全信息

• 海关编码: 2914509090

杜鹃黄素海关

• 海关编码: 2914509090
• 中文概述: 2914509090 含其他含氧基的酮. 增值税率:17.0% 退税率:9.0% 监管条件:无 最惠国关税:5.5% 普通关税:30.0%
• 申报要素: 品名, 成分含量, 用途, 丙酮报明包装
• Summary: HS:2914509090 other ketones with other oxygen function VAT:17.0% Tax rebate rate:9.0% Supervision conditions:none MFN tariff:5.5% General tariff:30.0%

杜鹃黄素靶点实验

查看更多实验

实验名称：Inhibition of NOX4 expressed in HEK293 FS cells at 10 uM assessed as H2O2 production ... 来源：ChEMBL 靶标：NADPH oxidase 4 External Id：CHEMBL1249160

实验名称：Cytotoxicity against human free style HEK293 cells after 72 hrs 来源：ChEMBL 靶标：HEK293 External Id：CHEMBL1249159

实验名称：Inhibition of NOX4 expressed in HEK293 FS cells assessed as H2O2 production by H2O2/T... 来源：ChEMBL 靶标：NADPH oxidase 4 External Id：CHEMBL1249158

实验名称：Inhibition of NOX4 expressed in HEK293 FS cells at 10 uM assessed as H2O2 production ... 来源：ChEMBL 靶标：NADPH oxidase 4 External Id：CHEMBL1249157

实验名称：Antioxidant activity assessed as DPPH free radical scavenging activity by measuring r... 来源：ChEMBL 靶标：N/A External Id：CHEMBL3862528

实验名称：Antioxidant activity assessed as DPPH free radical scavenging activity at 5 uM after ... 来源：ChEMBL 靶标：N/A External Id：CHEMBL3862529

实验名称：Enhancement of HSP27 Ser78 phosphorylation in human HeLa cells at 50 ug/mL treated fo... 来源：ChEMBL 靶标：Heat shock protein beta-1 External Id：CHEMBL993710

实验名称：Inhibition of heat-induced HSP70 expression in human Jurkat cells at 50 ug/mL treated... 来源：ChEMBL 靶标：Jurkat External Id：CHEMBL993709

实验名称：Inhibition of thrombin in New Zealand rabbit plasma assessed as activated partial thr... 来源：ChEMBL 靶标：Thrombin External Id：CHEMBL2045782

实验名称：Anticoagulant activity in rabbit plasma assessed as activated partial thromboplastin ... 来源：ChEMBL 靶标：Plasma External Id：CHEMBL5127306

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杜鹃黄素英文别名

• Quercetin 5-methyl ether
• 3,7,3',4'-tetrahydroxy-5-methoxyflavone
• 2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-5-methoxychromen-4-one
• Azaleatin
• 5-O-Methyl Quercetin