卡非多

• 常用名: 卡非多
• 英文名: Carphedon
• CAS号: 77472-70-9
• 分子量: 218.252
• 密度: 1.2±0.1 g/cm3
• 沸点: 486.4±45.0 °C at 760 mmHg
• 分子式: C₁₂H₁₄N₂O₂
• 熔点: N/A
• 闪点: 247.9±28.7 °C

卡非多用途

Phenylpiracetam(Phenotropyl; Phenotropil)是piracetam的苯基衍生物,活性较piracetam高30到60倍。

卡非多名称

• 中文名: 4-苯基-2-吡咯烷酮-1-乙酰胺
• 英文名: 2-(2-Oxo-4-phenylpyrrolidin-1-yl)acetamide
• 中文别名: 苯基吡拉西坦 | 芳妥西坦 | 4-苯基吡拉西坦 | 卡非多

卡非多生物活性

• 描述: Phenylpiracetam(Phenotropyl; Phenotropil)是piracetam的苯基衍生物,活性较piracetam高30到60倍。
• 相关类别:
  信号通路 >> 跨膜转运 >> GABA受体
  信号通路 >> 神经信号通路 >> GABA受体
  研究领域 >> 神经疾病
• 参考文献:

  [1]. Zvejniece L, et al. Investigation into stereoselective pharmacological activity of phenotropil. Basic Clin Pharmacol Toxicol. 2011 Nov;109(5):407-12.

卡非多物理化学性质

• 密度: 1.2±0.1 g/cm3
• 沸点: 486.4±45.0 °C at 760 mmHg
• 分子式: C₁₂H₁₄N₂O₂
• 分子量: 218.252
• 闪点: 247.9±28.7 °C
• 精确质量: 218.105530
• PSA: 64.39000
• LogP: 0.16
• InChIKey: LYONXVJRBWWGQO-UHFFFAOYSA-N
• SMILES: NC(=O)CN1CC(c2ccccc2)CC1=O
• 蒸汽压: 0.0±1.2 mmHg at 25°C
• 折射率: 1.580

卡非多毒性和生态

卡非多安全信息

• 海关编码: 2933990090

卡非多海关

• 海关编码: 2933990090
• 中文概述: 2933990090. 其他仅含氮杂原子的杂环化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%
• 申报要素: 品名, 成分含量, 用途, 乌洛托品请注明外观, 6－己内酰胺请注明外观, 签约日期
• Summary: 2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

卡非多靶点实验

查看更多实验

实验名称：Primary cell-based high-throughput screening assay for identification of compounds th... 来源：Johns Hopkins Ion Channel Center 靶标：regulator of G-protein signaling 4 isoform 2 [Homo sapiens] External Id：JHICC_RGS_Act_HTS

实验名称：Luminescence-based cell-based primary high throughput screening assay to identify ago... 来源：The Scripps Research Institute Molecular Screening Center 靶标：mu-type opioid receptor isoform MOR-1 [Homo sapiens] External Id：OPRM1-OPRD1_AG_LUMI_1536_1X%ACT PRUN

实验名称：QFRET-based biochemical primary high throughput screening assay to identify exosite i... 来源：The Scripps Research Institute Molecular Screening Center 靶标：disintegrin and metalloproteinase domain-containing protein 17 preproprotein [Homo sapiens] External Id：ADAM17_INH_QFRET_1536_1X%INH PRUN

实验名称：Fluorescence-based cell-based primary high throughput screening assay to identify ago... 来源：The Scripps Research Institute Molecular Screening Center 靶标：muscarinic acetylcholine receptor M1 [Homo sapiens] External Id：CHRM1_AG_FLUO8_1536_1X%ACT PRUN

实验名称：uHTS identification of small molecule activators of the adaptive arm of the Unfolded ... 来源：Burnham Center for Chemical Genomics 靶标：N/A External Id：BCCG-A405-UPR-XBP1-PrimaryAgonist-Assay

实验名称：High throughput fluorescence intensity-based biochemical assay to screen for small mo... 来源：University of Pittsburgh Molecular Library Screening Center 靶标：furin (paired basic amino acid cleaving enzyme), isoform CRA_a [Homo sapiens] External Id：MH080376 Biochemical HTS for Inhibitors of the Proprotein Convertase Furin.

实验名称：Fluorescence polarization to screen for inhibitor that competite the binding of FadD2... 来源：Broad Institute 靶标：FATTY-ACID-CoA LIGASE FADD28 (FATTY-ACID-CoA SYNTHETASE) External Id：2147-01_Inhibitor_SinglePoint_HTS_Activity

实验名称：Bursicon-induced LGR2 mediated cAMP production in LGR-2/CRE6x-Luciferase co-transfect... 来源：Broad Institute 靶标：N/A External Id：Bursicon-induced LGR2 mediated cAMP production in LGR-2/CRE6x-Luciferase co-transfected HEK293 cells Inhibition - 7011-01_Antagonist_SinglePoint_HTS_Activity

实验名称：Fluorescence-based cell-based primary high throughput screening assay to identify pos... 来源：The Scripps Research Institute Molecular Screening Center 靶标：muscarinic acetylcholine receptor M1 [Homo sapiens] External Id：CHRM1_PAM_FLUO8_1536_1X%ACT PRUN

实验名称：Fluorescence polarization-based biochemical high throughput primary assay to identify... 来源：The Scripps Research Institute Molecular Screening Center 靶标：RecName: Full=Sialate O-acetylesterase; AltName: Full=H-Lse; AltName: Full=Sialic acid-specific 9-O-acetylesterase; Flags: Precursor [Homo sapiens] External Id：SIAE_INH_FP_1536_1X%INH PRUN

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卡非多英文别名

• fonturacetam
• UNII:99QW5JU66Y
• Carphedon
• Phenylpiracetam
• 4-Phenyl-2-pyrrolidone-1-acetamide
• 2-(2-Oxo-4-phenyl-1-pyrrolidinyl)acetamide
• 2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
• 4-Phenylpiracetam
• Phenotropil