6BrCaQ

• 常用名: 6BrCaQ
• 英文名: 6BrCaQ
• CAS号: 954416-67-2
• 分子量: 387.23
• 密度: N/A
• 沸点: N/A
• 分子式: C₁₈H₁₅BrN₂O₃
• 熔点: N/A
• 闪点: N/A

6BrCaQ用途

6BrCaQ是一种有效的线粒体热休克蛋白TRAP1抑制剂,具有抗增殖活性。6BrCaQ可用于合成6BrCaQ TPP共轭物[1]。

6BrCaQ名称

• 英文名: 6BrCaQ

6BrCaQ生物活性

• 描述: 6BrCaQ是一种有效的线粒体热休克蛋白TRAP1抑制剂,具有抗增殖活性。6BrCaQ可用于合成6BrCaQ TPP共轭物[1]。
• 相关类别:
  研究领域 >> 癌症
  信号通路 >> 代谢酶/蛋白酶 >> HSP
  信号通路 >> 细胞周期/DNA损伤 >> HSP
• 参考文献:

  [1]. Mathieu C, et, al. Synthesis and antiproliferative activity of 6BrCaQ-TPP conjugates for targeting the mitochondrial heat shock protein TRAP1. Eur J Med Chem. 2022 Feb 5;229:114052.

6BrCaQ物理化学性质

• 分子式: C₁₈H₁₅BrN₂O₃
• 分子量: 387.23
• InChIKey: RCKMJRZPGJEVGF-UHFFFAOYSA-N
• SMILES: COc1ccc(C(=O)Nc2cc3cc(Br)ccc3n(C)c2=O)cc1

6BrCaQ靶点实验

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