1-Allyl-3,7-dimethyl-8-p-sulfophenylxanthine Sodium Salt

1-Allyl-3,7-dimethyl-8-p-sulfophenylxanthine Sodium Salt Structure
1-Allyl-3,7-dimethyl-8-p-sulfophenylxanthine Sodium Salt structure
Common Name 1-Allyl-3,7-dimethyl-8-p-sulfophenylxanthine Sodium Salt
CAS Number 149981-25-9 Molecular Weight 376.38700
Density 1.49 g/cm3 Boiling Point N/A
Molecular Formula C16H16N4O5S Melting Point >300ºC
MSDS Chinese USA Flash Point N/A

Effect of trifluoromethyl and other substituents on activity of xanthines at adenosine receptors.

J. Med. Chem. 38 , 2639, (1993)

An aryl p-(trifluoromethyl) substituent increases the affinity of 1,3-disubstituted 8-phenylxanthines at A2a-adenosine receptors, while having little effect on affinity at A1-adenosine receptors. In contrast, an aryl p-(trifluoromethyl) substituent has little...

Functional coupling of human adenosine receptors to a ligand-dependent reporter gene system.

Biochem. Biophys. Res. Commun. 198 , 626, (1994)

We have stably transfected CHO cells that have integrated in their genome a reporter gene under the control of promoter sequences containing several copies of the cAMP response element, CRE, with different human adenosine receptors: A1, A2a and A2b. The new c...