Epiamastatin · HCl

Epiamastatin · HCl Structure
Epiamastatin · HCl structure
Common Name Epiamastatin · HCl
CAS Number 100992-59-4 Molecular Weight 511.00900
Density N/A Boiling Point 808ºC at 760mmHg
Molecular Formula C21H39ClN4O8 Melting Point N/A
MSDS Chinese USA Flash Point 442.5ºC

Inhibition of aminopeptidases by amastatin and bestatin derivatives. Effect of inhibitor structure on slow-binding processes.

J. Med. Chem. 27 , 417, (1984)

Amastatin [(2S,3R)-3-amino-2-hydroxy-5-methylhexanoyl-L-valyl-L-valyl-L- aspartic acid] and bestatin [(2S,3R)-3-amino-2-hydroxy-4-phenylbutanoyl-L-leucine] are slow-binding, competitive inhibitors of aminopeptidase M (AP-M) with net inhibition constants (Ki) ...