e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521

Compounds with antiulcer and antisecretory activity. II: 3-Heteroaryl-benzimidazolin-2-ones

M Bianchi, A Butti, S Rossi, F Barzaghi…

Index: Bianchi; Butti; Rossi; et al. European Journal of Medicinal Chemistry, 1983 , vol. 18, # 6 p. 495 - 500

Full Text: HTML

Citation Number: 6

Abstract

... II: 3-Heteroaryl-benzimidazolin-2-ones. Auteur(s) / Author(s). BIANCHI M. ; BUTTI A. ; ROSSI S. ; BARZAGHI F. ; MARCARIA V. ; Affiliation(s) du ou des auteurs / Author(s) Affiliation(s). Univ. Milano, ist. chimica farmaceutica Résumé / Abstract. Synthèse, relation structure-activité, toxicité Revue / Journal Title. European journal of medicinal chemistry ISSN 0223-5234 CODEN EJMCA5 Source / Source. 1983, vol. 18, n o 6, pp. 495-500 (9 ref.) Langue / Language. ...

2-Chloropyrazine Structure

2-Chloropyrazine

2H-Benzimidazol-2-one,5-chloro-1-ethyl-1,3-dihydro-(9CI) Structure

2H-Benzimidazol...

~33%

5-chloro-1-ethyl-3-pyrazin-2-ylbenzimidazol-2-one Structure

5-chloro-1-ethy...

3-Bromothiophene Structure

3-Bromothiophene

2H-Benzimidazol-2-one,5-chloro-1,3-dihydro-1-methyl-(9CI) Structure

2H-Benzimidazol...

~12%

5-chloro-1-methyl-3-thiophen-3-ylbenzimidazol-2-one Structure

5-chloro-1-meth...

6-chloro-3-methyl-2-oxobenzimidazole-1-carbonitrile Structure

6-chloro-3-meth...

~47%

5-chloro-1-methyl-3-(2H-tetrazol-5-yl)benzimidazol-2-one Structure

5-chloro-1-meth...

2H-Benzimidazol-2-one,5-chloro-1,3-dihydro-1-methyl-(9CI) Structure

2H-Benzimidazol...

~%

5-chloro-1-methyl-3-(2H-tetrazol-5-yl)benzimidazol-2-one Structure

5-chloro-1-meth...

2-Amino-6-picoline Structure

2-Amino-6-picoline

1-Chloro-3,4-dinitrobenzene Structure

1-Chloro-3,4-di...

~44%

N-(5-chloro-2-nitrophenyl)-6-methylpyridin-2-amine Structure

N-(5-chloro-2-n...

4-Chloro-N-methyl-2-nitroaniline Structure

4-Chloro-N-meth...

Ethyl chloroformate Structure

Ethyl chloroformate

~84%

ethyl N-[(5-chloro-2-nitrophenyl)methyl]carbamate Structure

ethyl N-[(5-chl...

ethyl N-[(4-chloro-2-nitrophenyl)methyl]carbamate Structure

ethyl N-[(4-chl...

~67%

ethyl N-[(2-amino-4-chlorophenyl)methyl]carbamate Structure

ethyl N-[(2-ami...

ethyl N-[(5-chloro-2-nitrophenyl)methyl]carbamate Structure

ethyl N-[(5-chl...

~83%

ethyl N-[(2-amino-5-chlorophenyl)methyl]carbamate Structure

ethyl N-[(2-ami...

N1-Ethylbenzene-1,2-diamine Structure

N1-Ethylbenzene...

Ethyl chloroformate Structure

Ethyl chloroformate

~9%

ethyl N-[2-(ethylamino)phenyl]carbamate Structure

ethyl N-[2-(eth...

ethyl N-[2-[2-(ethoxycarbonylamino)ethyl]phenyl]carbamate Structure

ethyl N-[2-[2-(...

N1-Ethylbenzene-1,2-diamine Structure

N1-Ethylbenzene...

Ethyl chloroformate Structure

Ethyl chloroformate

~12%

ethyl N-[2-(ethylamino)phenyl]carbamate Structure

ethyl N-[2-(eth...

ethyl N-[2-[2-(ethoxycarbonylamino)ethyl]phenyl]carbamate Structure

ethyl N-[2-[2-(...

N1-ISOPROPYL-4-CHLORO-2-NITROANILINE Structure

N1-ISOPROPYL-4-...

~%

ethyl N-[5-chloro-2-(propan-2-ylamino)phenyl]carbamate Structure

ethyl N-[5-chlo...

1,4-Dichloro-2-nitrobenzene Structure

1,4-Dichloro-2-...

~%

ethyl N-[5-chloro-2-(propan-2-ylamino)phenyl]carbamate Structure

ethyl N-[5-chlo...

Ethyl chloroformate Structure

Ethyl chloroformate

5-CHLORO-2-(ISOPROPYLAMINO)ANILINE Structure

5-CHLORO-2-(ISO...

~42%

ethyl N-[5-chloro-2-(propan-2-ylamino)phenyl]carbamate Structure

ethyl N-[5-chlo...

N-(5-chloro-2-nitrophenyl)pyridin-2-amine Structure

N-(5-chloro-2-n...

~%

ethyl N-[4-chloro-2-(pyridin-2-ylamino)phenyl]carbamate Structure

ethyl N-[4-chlo...

Ethyl chloroformate Structure

Ethyl chloroformate

N/A Structure

~77%

ethyl N-[4-chloro-2-(pyridin-2-ylamino)phenyl]carbamate Structure

ethyl N-[4-chlo...

5-CHLORO-2-(ISOPROPYLAMINO)ANILINE Structure

5-CHLORO-2-(ISO...

~%

6-chloro-3-propan-2-yl-1H-benzimidazol-2-one Structure

6-chloro-3-prop...

ethyl N-[5-chloro-2-(propan-2-ylamino)phenyl]carbamate Structure

ethyl N-[5-chlo...

~78%

6-chloro-3-propan-2-yl-1H-benzimidazol-2-one Structure

6-chloro-3-prop...

isopropylamine Structure

1,4-Dichloro-2-nitrobenzene Structure

1,4-Dichloro-2-...

~70%

N1-ISOPROPYL-4-CHLORO-2-NITROANILINE Structure

N1-ISOPROPYL-4-...

Cyanogen bromide Structure

Cyanogen bromide

2H-Benzimidazol-2-one,5-chloro-1,3-dihydro-1-methyl-(9CI) Structure

2H-Benzimidazol...

~71%

6-chloro-3-methyl-2-oxobenzimidazole-1-carbonitrile Structure

6-chloro-3-meth...

5-Chloro-2-nitro-N-methylaniline Structure

5-Chloro-2-nitr...

Ethyl chloroformate Structure

Ethyl chloroformate

~%

ethyl N-[(4-chloro-2-nitrophenyl)methyl]carbamate Structure

ethyl N-[(4-chl...