GSK2973980A

Modify Date: 2024-01-05 16:58:37

GSK2973980A Structure
GSK2973980A structure
Common Name GSK2973980A
CAS Number 2219321-25-0 Molecular Weight 534.43
Density N/A Boiling Point N/A
Molecular Formula C25H19F5N4O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of GSK2973980A


GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.

 Names

Name GSK2973980A

 GSK2973980A Biological Activity

Description GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.
Related Catalog
Target

IC50: 3 nM (DGAT1)[1]

References

[1]. Cheung M, et al. Discovery of Tetralones as Potent and Selective Inhibitors of Acyl-CoA:Diacylglycerol Acyltransferase 1. ACS Med Chem Lett. 2018 Jan 16;9(2):103-108.

 Chemical & Physical Properties

Molecular Formula C25H19F5N4O4
Molecular Weight 534.43
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