Name | ZXH-3-26 |
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Description | ZXH-3-26 is a selective BRD4 degrader with a DC50/5h (DC50/5h referring to half-maximal degradation after 5 hours of treatment) of ~ 5 nM[1]. |
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Related Catalog | |
Target |
BRD4:5 nM (DC50, 5 hours of treatment) |
In Vitro | ZXH-3-26 represents the first small molecule to allow pharmacologic targeting of BRD4 without significant inhibition or degradation of BRD2/3[1]. |
References |
Molecular Formula | C38H37ClN8O7S |
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Molecular Weight | 785.27 |
Hazard Codes | Xi |
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