2235358-74-2

2235358-74-2 structure

Name: Deltasonamide 2 (TFA)
Chemical Name: Deltasonamide 2 TFA
CAS Number: 2235358-74-2
Molecular Formula: C₃₂H₄₀ClF₃N₆O₆S₂
Molecular Weight: 761.27
Catalog: Signaling Pathways Metabolic Enzyme/Protease Phosphodiesterase (PDE)
Create Date: 2019-06-30 16:59:15
Modify Date: 2024-01-10 11:21:24
Deltasonamide 2 TFA is a PDEδ inhibitor with a Kd of ~385 pM and an EC50 of 1.24 μM[1].

Name	Deltasonamide 2 TFA

Description	Deltasonamide 2 TFA is a PDEδ inhibitor with a Kd of ~385 pM and an EC50 of 1.24 μM[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Metabolic Enzyme/Protease >> Phosphodiesterase (PDE)
Target	Kd: ~385 pM (PDEδ)[1] EC50: 1.24 ± 0.06 μM (PDEδ)[1]
References	[1]. Klein CH, et al. PDEδ inhibition impedes the proliferation and survival of human colorectal cancer cell linesharboring oncogenic KRas. Int J Cancer. 2019 Feb 15;144(4):767-776.