Name | CBP bromodomain inhibitor |
---|
Description | a potent, selective CBP bromodomain inhibitor with IC50 of 69 nM, displays exquisite selectivity over BRD4(1) (IC50=18 uM) and the broader bromodomain family. |
---|---|
References | References 1. Bronner SM, et al. J Med Chem. 2017 Dec 28;60(24):10151-10171. View Related Products by Target Bromodomain |
Molecular Formula | C22H20F2N4OS |
---|---|
Molecular Weight | 426.486 |