Name | Bromodomain inhibitor-10 |
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Description | Bromodomain inhibitor-10 (compound 128) is a potent bromodomain inhibitor with Kds of 15.0, 2500 nM for BRD4-1 and BRD4-2, respectively. Bromodomain inhibitor-10 inhibits the production of IL12p40[1]. |
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Related Catalog | |
Target |
BRD4-1:15 nM (Kd) BRD4-2:2500 nM (Kd) |
References |
[1]. Jimmi GERNER SEITZBERG, et al. Compounds active towards bromodomains. WO2016016316A1 |
Molecular Formula | C20H20N4O3 |
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Molecular Weight | 364.40 |