1870849-58-3

1870849-58-3 structure
1870849-58-3 structure
  • Name: Bromodomain inhibitor-10
  • Chemical Name: Bromodomain inhibitor-10
  • CAS Number: 1870849-58-3
  • Molecular Formula: C20H20N4O3
  • Molecular Weight: 364.40
  • Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
  • Create Date: 2022-09-01 11:45:16
  • Modify Date: 2024-01-23 14:00:09
  • Bromodomain inhibitor-10 (compound 128) is a potent bromodomain inhibitor with Kds of 15.0, 2500 nM for BRD4-1 and BRD4-2, respectively. Bromodomain inhibitor-10 inhibits the production of IL12p40[1].

Name Bromodomain inhibitor-10
Description Bromodomain inhibitor-10 (compound 128) is a potent bromodomain inhibitor with Kds of 15.0, 2500 nM for BRD4-1 and BRD4-2, respectively. Bromodomain inhibitor-10 inhibits the production of IL12p40[1].
Related Catalog
Target

BRD4-1:15 nM (Kd)

BRD4-2:2500 nM (Kd)

References

[1]. Jimmi GERNER SEITZBERG, et al. Compounds active towards bromodomains. WO2016016316A1

Molecular Formula C20H20N4O3
Molecular Weight 364.40