Name | PF-06678419 |
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Description | PF-06678419 (PF06678419) is a potent, selective inhibitor of the Na+/citrate transporter NaCT (SLC13A5) that shows inhibition of citrate uptake in the HEKNaCT cells with IC50 of 0.44 uM; displays relatively selectivity over NaDC1 and NaDC3 (7-10-fold). |
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References | References 1. Pajor AM, et al. Mol Pharmacol. 2016 Dec;90(6):755-765. 2. Huard K, et al. Sci Rep. 2015 Dec 1;5:17391. View Related Products by Target Sodium-coupled Citrate Transporter (NaCT,SLC13A5) |
Molecular Formula | C12H13IO5 |
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Molecular Weight | 364.135 |