Name | YAP-TEAD-IN-1 TFA |
---|
Description | YAP-TEAD-IN-1 TFA is a potent and competitive peptide inhibitor of YAP-TEAD interaction (IC50=25 nM). YAP-TEAD-IN-1 TFA is a 17mer peptide and shows a higher the binding affinity to TEAD1 (Kd=15 nM) than YAP (50-171) (Kd= 40 nM)[1]. |
---|---|
Related Catalog | |
Target |
IC50: 25 nM (YAP-TEAD interaction)[1] |
In Vitro | YAP-TEAD-IN-1 (peptide 17)(2 μM) is against endogenous YAP binding to GST-TEAD(1209-426) in a GST pull-down assay, the Kd of His-YAP(1209-426) is determined to be 40 nM[1]. |
References |
Molecular Formula | C93H144ClN23O21S2.xC2HF3O2 |
---|